Browsing by Author CHEONG SIEW LEE

Showing results 1 to 8 of 8
Issue DateTitleAuthor(s)
2015A facile and novel synthesis of N2-, C6-substituted pyrazolo[3,4- d ]pyrimidine-4 carboxylate derivatives as adenosine receptor antagonistsVenkatesan G. ; Paira P.; Cheong S.L. ; Federico S.; Klotz K.N.; Spalluto G.; Pastorin G. 
1-Jan-2011Biomedical applications I: Delivery of drugsSpalluto, G.; Federico, S.; Cacciari, B.; Bianco, A.; Cheong, S.L. ; Prato, M.
15-Oct-2011Does the combination of optimal substitutions at the C 2-, N 5- and N 8-positions of the pyrazolo-triazolo-pyrimidine scaffold guarantee selective modulation of the human A 3 adenosine receptors?Cheong, S.L. ; Dolzhenko, A.V. ; Paoletta, S.; Lee, E.P.R.; Kachler, S.; Federico, S.; Klotz, K.-N.; Dolzhenko, A.V. ; Spalluto, G.; Moro, S.; Pastorin, G. 
17-Jun-2013Organoruthenium antagonists of human A3 adenosine receptorsPaira, P. ; Chow, M.J.; Venkatesan, G.; Kosaraju, V.K.; Cheong, S.L. ; Klotz, K.-N.; Ang, W.H. ; Pastorin, G. 
15-May-2011Pharmacophore elucidation for a new series of 2-aryl-pyrazolo-triazolo- pyrimidines as potent human A3 adenosine receptor antagonistsCheong, S.L. ; Federico, S.; Venkatesan, G.; Paira, P. ; Shao, Y.-M.; Spalluto, G.; Yap, C.W. ; Pastorin, G. 
10-Feb-2011Synthesis and biological evaluation of a new series of 1, 2, 4-triazolo[1, 5-α]-1, 3, 5-triazines as human a 2a adenosine receptor antagonists with improved water solubilityFederico, S.; Paoletta, S.; Cheong, S.L. ; Pastorin, G. ; Cacciari, B.; Stragliotto, S.; Norbert Klotz, K.; Siegel, J.; Gao, Z.-G.; Jacobson, K.A.; Moro, S.; Spalluto, G.
Mar-2013The A3 adenosine receptor as multifaceted therapeutic target: Pharmacology, medicinal chemistry, and in silico approachesCheong, S.L. ; Federico, S.; Venkatesan, G.; Mandel, A.L. ; Shao, Y.-M.; Moro, S.; Spalluto, G.; Pastorin, G. 
22-Apr-2010The significance of 2-furyl ring substitution with a 2-(para -substituted) aryl group in a new series of pyrazolo-triazolo-pyrimidines as potent and highly selective hA3 adenosine receptors antagonists: New insights into structure-affinity relationship and receptor-antagonist recognitionCheong, S.L. ; Dolzhenko, A. ; Kachler, S.; Paoletta, S.; Federico, S.; Cacciari, B.; Dolzhenko, A. ; Klotz, K.-N.; Moro, S.; Spalluto, G.; Pastorin, G.